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Liotta, Dennis C, Emory University
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Investigation and Modeling of Binding Modes of Novel Small-Molecule Nox2 Inhibitors
Chapter 1. Total synthesis of Fumonisin B1 Chapter 2. Synthesis of Unnatural Sphingoli...
Design, Synthesis, and Biological Evaluation of Subunit Selective N-Methyl-D-Aspartate...
I. A New Approach to the Synthesis of a Key 5-Oxo-Pyridinyl Molybdenum Scaffold. II. O...
Identification of Small Molecule Inhibitors of I-κB Kinase
Expanding the Scope of Donor/Acceptor Carbenes and the Synthesis of Novel Therapeutic ...
Part I: Synthesis of Cyclobutyl Nucleoside Analogs That Mimic AZT for Inhibition of th...
Incorporating the Scientific Contributions of Research Faculty into the Chemical Educa...
Development of a Copper Catalyzed Aminoacetoxylation Reaction of Olefins, Development ...
Chapter 1: The development of a model system for the B-ring of brevenal and methods fo...
Synthesis of 2'-Fluoro-2',3'-Dideoxynucleosides as Inhibitors of Hepatitis...
Investigation of C-H Bond Oxidation Reactions: I. Asymmetric Amination of C-H Bonds Us...
Use of Receptor-Based Drug Design and Applications in the Study of finding antagonists...
Progress Toward the Total Synthesis of PM-toxin A And Future Development of Mild Lewis...
Screening, hit expansion and mechanistic studies for natural product analogs derived f...
Development of Monocarbonyl Curcumin Analogues Towards Treating Tuberculosis and Cancer
SYNTHESIS OF CYCLOPROPANES AND DIHYDROFURANS BY METAL CARBENOID REACTIONS
Part I: Design, Synthesis, and Biological Activity of NMDA Receptor Antagonists Part I...
Validation of Receptor-Based Drug Design and Applications in the Study of IKKs, Trunca...
Inhibition of the NF-κB signaling pathway by the curcumin analogs, 3,5-Bis(2-pyridinyl...
Rhodium Alkenylcarbenes: Novel Reactivity and Precursors
Progress Toward a Common Intermediate for C1 Modified Enigmols
Design, Synthesis, and Biological Evaluation of Subunit-Selective N-Methyl-D-Aspartate...
Tumor Necrosis Factor-alpha mediated transactivation of the Epidermal Growth Factor Re...
Structural Determinants of Activity, Mechanism and Structure Activity Relationships of...
ASYMMETRIC REACTIONS OF DONOR/ACCEPTOR RHODIUM CARBENOIDS: FROM FORMAL CYCLOADDITIONS ...
Organometallic Enantiomeric Scaffolds in the Synthesis of Alkaloids: I. Homo-SN2´-like...
Design, Synthesis, and Biologic Evaluation of Tetrahydroisoquinoline-Based CXCR4 Modul...
Design, Synthesis, and Biological Evaluation of Subunit-Selective N-Methyl-D-Aspartate...
Application of fluorescent nucleoside analogs in direct evolution of Drosophila melano...
Generating designer enzymes for therapeutic and industrial applications
Navigating the Roads to Drug Discovery: Part 1: Design, Synthesis, and Biological Eval...
Design, Synthesis and Biological Evaluation of C4-C9 Bridged Epothilone Analogs
Computer-Assisted Drug Discovery Part I: Design, Development, Validation and Applicati...
Incorporating Transition Metal Organometallic Chemistry into the Introductory Organic ...
Synthetic Studies Toward Cyclobutyl Nucleoside Analogs for the Treatment of Hepatitis ...
Towards the Development of Non-Toxic Therapeutics in the Fight Against Cancer
Optimization of Dual-tropic CXCR4/CCR5 HIV-1 Entry Inhibitors and a Market Analysis
Development of a novel stereo-selective synthetic route towards Pumiliotoxin C, potent...
Part I. Design of a novel class of reversible non-covalent small molecule inhibitors f...
SYNTHESIS OF SMALL MOLECULE THERAPEUTICS UTILIZING RHODIUM CARBENOID CHEMISTRY
Multi-mechanism antiretroviral approach targeting macrophage derived viral sanctuaries
Design, Development and Application of a Novel In-Silico High-throughput Screening App...
Potential Cross-Talk between the Aryl Hydrocarbon Receptor (AHR) and the Constitutive ...
Use of Furans as Vehicles for Heterocyclic Synthesis: Anaza-Achmatowicz Approach to Pi...
Part I: Design, Synthesis and Biological Evaluation of C6-C8 Bridged Epothilone Analog...
Engineering The Substrate Specificity Of Human Deoxycytidine Kinase
Synthesis and Characterization of Unusal Amphiphiles Part I. Nonsteroidal Facial Amph...
Part 1: Stereoselective Synthesis of Quaternary Center BearingAzetines and β-Amino Aci...
Synthesis of Those Sectors of Saccharomicin A and B ContainingSaccharosamine and the D...
Computational Studies of Ligand Protein Interactions Part I: TheT-Taxol Conformation P...
Part I: Conformational Analysis of Bioactive Molecules inSolutionPart II: Structure-Ba...
Synthesis of Altromycin and Kidamycin Aglycones from a Common Intermediate & Studi...
Metal Mediated Cross-Coupling Reactions for Carbon-Carbon andCarbon-Nitrogen Bonds For...
Part I: Synthesis of Cyclobutyl Nucleoside and NucleotideAnalogues as HIV-1 Reverse Tr...
Synthesis and Anti-Viral Activity of Novel 3,6-dioxa-[3.2.0]bicyclonucleoside Nucleoti...
Part I: Structure and Function in the NMDA Ligand Binding DomainPart II: Comparison of...
Analysis of the EF24-modulated signaling pathways for thedevelopment of novel cancer c...
Towards the Synthesis of Marine Polyether Triterpenes
Paclitaxel and Cyclostreptin in theTubulin Binding Site
Part 1: Synthesis and Anti-HIV Activity of Novel CyclobutylNucleoside and Nucleotide A...
Part I: Measles virus entry into cells and the inhibition offusion and replicationPart...
Development of Fluorescence-based Molecular Tension Probes to Investigate Cellular Mec...
Discovery and Synthesis of Next Generation Chemokine Modulators with or without Concur...
Part 1. Discovery of a Fluorinated Enigmol Analog with Enhanced Pharmacokinetic and An...
Acylative Redox Dehydration of Carboxylic Acids and Benzoisothiazolones in the Synthes...
The Design, Synthesis, and Biological Evaluation of Subunit-selective N-Methyl-D-Aspar...
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2012
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2008
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School
Laney Graduate School
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Emory College
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Department
Chemistry
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Biological and Biomedical Sciences
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PhD
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MS
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Dissertation
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Master's Thesis
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Chemistry, Organic
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Committee
Liotta, Dennis C, Emory University
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67
McDonald, Frank, Emory University
17
Liebeskind, Lanny S, Emory University
16
Blakey, Simon, Emory University
14
Lynn, David, Emory University
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HIV
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CXCR4
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cancer
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nucleoside
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Conformation
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