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Design, Development and Application of a Novel In-Silico
High-throughput Screening Approach
1 di 10
SYNTHESIS OF SMALL MOLECULE THERAPEUTICS UTILIZING RHODIUM
CARBENOID CHEMISTRY
2 di 10
Towards the Development of Non-Toxic Therapeutics in the Fight
Against Cancer
3 di 10
Part I: Design, Synthesis and Biological Evaluation of C6-C8 Bridged Epothilone AnalogsPart II: Discovery of Small Molecule CXCR4 Antagonists
4 di 10
Computer-Assisted Drug Discovery Part I: Design, Development,
Validation and Application of FRESH, a Novel In-Silico
High-throughput Screening Program Part II: Monocarbonyl Curcumin
Analogues: Heterocyclic Pleiotropic Kinase Inhibitors that Mediate
Anticancer Properties Part III: Development of 2nd Generation
NAMFIS Software Program by Java
5 di 10
Progress Toward a Common Intermediate for C1 Modified
Enigmols
6 di 10
Synthesis of Ellagic Acid Glycoside Derivatives found in Rubus
ulmifolius
7 di 10
Design, Synthesis, and Biological Evaluation of Subunit-Selective
N-Methyl-D-Aspartate Receptor Antagonists
8 di 10
Part I: Conformational Analysis of Bioactive Molecules inSolutionPart II: Structure-Based Design of Selective Inhibitors ofCyclin-Dependent Kinase 7
9 di 10
Aerobic, Medal Mediated Ketone Synthesis from Thiol Esters and Boronic Acids
10 di 10