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The Development of VIP Antagonist (ANT) Peptide Derivatives and Synthetic Approaches towards the Ryptide Macrocycle
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Designing a Library of Conjugated Planar Chiral Rh(III) Indenyl Catalysts and Progress Towards an Enantioselective Intramolecular 1,2-Arylamination of Terminal Olefins using Planar Chiral Rh(III) Indenyl Catalysts
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Optimization and Investigation of a Photoredox-Driven Selective Radical Cyclization
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Understanding the Reactivity of Planar Chiral Naphthindenyl Rhodium(III) Catalysts
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Six Amino Acids: Accessing OAS1 Inhibitors
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Synthesis of P1 and Cap-P2 Fragments of Novel SARS-CoV-2 Protease Inhibitors
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Total Synthesis and Target Identification of Pestalachloride B to Facilitate Antibiotic Development
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Synthetic Investigations Into the Diterpenoids Larikaempferic Methyl Ester and (-)-Hardwickiic Acid
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The Stereochemical Effect of HFIP on Asymmetric Rhodium(II)-Catalyzed Cyclopropanation
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Synthesis of Lipid Prodrugs of Tenofovir to Promote Lymphatic Uptake and Combat Toxicity
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Development of Enantioselective C–N Bond Forming Reactions using Planar Chiral Rh(III) Indenyl Catalysts
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Expanding the Toolbox: Development of Novel Chemical Tools for Profiling of Proteins and Dimethyl Post-translational Modification
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Systems Chemistry of Self-Replicating Networks: From Nature to Nanomaterials
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Structure-Activity Relationship Studies of EP2 Antagonists for Aqueous Solubility Enhancement
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Towards Ideal Synthesis: Concise Total Syntheses of Sesquiterpene and Diterpene Natural Products
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Fighting the Good Fight: Structure Based Design and Biological Investigation of Allosteric OAS1 Inhibitors for Mitigating Inborn Errors of Immunity
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Diagnostic Tools: Molecular Probes for the Detection of Biological Aldehydes
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A Generalized Approach to Deliver Functionalized Isoindolines in Macrocycles
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Developing Transition Metal Catalysts that Incorporate Redox-Active Ligand Frameworks for Sustainable Catalysis
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Development of New Diaryl Diazo Compounds and the Study of their application in C-H Functionalization Chemistry
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Development of New Diaryl Diazo Compounds and the Study of their application in C-H Functionalization Chemistry
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DNA mechanocapsules: Force responsive tetrahedral DNA nanostructures with modular cargo delivery for targeting mechanical phenotypes of diseases
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Metal Catalyst Methodology Development towards Carbon-Oxygen Bond Formation: Synthesis of Vinyl Ethers and Vinyl Esters
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The Development of Planar Chiral Indenyl Catalysts and the Progress Towards Synthesis of the Western Macrocycle of Darobactin A
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Group IX Metal-Catalyzed C–H Activation Towards the Development of New Synthetic Strategies
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Natural Product Inspired Complementary Approaches to Counter Antimicrobial Resistance: Synthetic and Biological Investigations of Antibacterial Small Molecules
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An Investigation on the Diastereoselectivity of α-Methylstyrene Cyclopropanations Catalyzed by Dirhodium (II) Catalysts
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Synthesis of Novel Nucleotide Tenofovir/Lamivudine Prodrug Conjugates for treatment of Human Immunodeficiency Virus and Hepatitis B
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Synthesis and Evaluation of Novel Phenyl-Adamantane Dirhodium Catalyst for C-H Functionalization
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New Advances in Asymmetric Cyclopropanation and Drug Discoveries Using Dirhodium(II) Tetracarboxylates
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Asparagine and Glutamine Bioconjugation
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Synthesis of alkyl analogues of 1,4-dihydropyridine for developing novel treatment against chemoresistance in prostate cancer
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Carboxylation of C(sp2) Bromides Enabled by Metallophotoredox Dual Catalysis and Sodium Formate
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Computational Modeling of Oxyradical and Metal-Oxo Reactivity and Selectivity in Hydrogen Atom Transfer Reactions
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Triazene Coarctate Cyclization for the Synthesis of Fluorescent Cyclic Peptides
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Overcoming Antibacterial Resistance through Synthesis of Small Molecules Targeting Efflux Mechanisms
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Overcoming the Limitations of Rhodium-Catalyzed Asymmetric Cyclopropanation and Other Adventures in Strained Ring Synthesis
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Catalytic Process for Epoxide Ring-Opening with Terminal Alkynes for Carbon-Carbon Bond Formation
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Novel Quaternary Ammonium Compounds Derived from the Antimicrobial Natural Product Ianthelliformisamine C
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Cu- and Pd-Catalyzed a-Hydroxycyclopropanol Ring Opening Reactions: Electrophilic Trappings to 3-Furanones, and Carbonylation to 4-Ketovalerolactones.
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Radical Reactivity via Transient Carbon Dioxide Radical Anion (CO2•−)
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Design and Synthesis of Chemical Modulators for Altered Activity of Nuclear Receptor Liver Receptor Homolog-1 and Synthesis of Spirocyclic Piperidines via Radical Hydroarylation
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Chemo and Site Selective Modification of Proteins and Chemical Tools for Studying Mono-Methyl Lysine (Kme)
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Developing Chemical Tools for Selective Peptide Modification
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Studies in Small Molecule Drug Discovery: Part I. Synthesis of Novel Nucleoside-Based Antivirals to Treat Hepatitis C; Part II. Validation and Implementation of a Machine Learning Algorithm to Create a Safer Kinase Inhibitor as a Potential First-in-Class Antiparkinsonian Agent
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Membranes & Metals: Bacterial Targets to Fight Antibiotic Resistance
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Exploration of Bilingual Peptide Nucleic Acids
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Development of Chemical Methods for Labeling Monomethyl Lysine Post-Translational Modification and Serine and their Applications.
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A Three-Pronged Approach to Combatting Antibiotic Resistance
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Synthesis and Biological Investigation of Membrane-targeting Antimicrobials
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