Search Constraints
« Previous |
1 - 100 of 241
|
Next »
Search Results
Select an image to start the slideshow
The Development of VIP Antagonist (ANT) Peptide Derivatives and Synthetic Approaches towards the Ryptide Macrocycle
1 of 100
Designing a Library of Conjugated Planar Chiral Rh(III) Indenyl Catalysts and Progress Towards an Enantioselective Intramolecular 1,2-Arylamination of Terminal Olefins using Planar Chiral Rh(III) Indenyl Catalysts
2 of 100
Optimization and Investigation of a Photoredox-Driven Selective Radical Cyclization
3 of 100
Understanding the Reactivity of Planar Chiral Naphthindenyl Rhodium(III) Catalysts
4 of 100
Six Amino Acids: Accessing OAS1 Inhibitors
5 of 100
Synthesis of P1 and Cap-P2 Fragments of Novel SARS-CoV-2 Protease Inhibitors
6 of 100
Total Synthesis and Target Identification of Pestalachloride B to Facilitate Antibiotic Development
7 of 100
Synthetic Investigations Into the Diterpenoids Larikaempferic Methyl Ester and (-)-Hardwickiic Acid
8 of 100
The Stereochemical Effect of HFIP on Asymmetric Rhodium(II)-Catalyzed Cyclopropanation
9 of 100
Synthesis of Lipid Prodrugs of Tenofovir to Promote Lymphatic Uptake and Combat Toxicity
10 of 100
Development of Enantioselective C–N Bond Forming Reactions using Planar Chiral Rh(III) Indenyl Catalysts
11 of 100
Expanding the Toolbox: Development of Novel Chemical Tools for Profiling of Proteins and Dimethyl Post-translational Modification
12 of 100
Systems Chemistry of Self-Replicating Networks: From Nature to Nanomaterials
13 of 100
Structure-Activity Relationship Studies of EP2 Antagonists for Aqueous Solubility Enhancement
14 of 100
Towards Ideal Synthesis: Concise Total Syntheses of Sesquiterpene and Diterpene Natural Products
15 of 100
Fighting the Good Fight: Structure Based Design and Biological Investigation of Allosteric OAS1 Inhibitors for Mitigating Inborn Errors of Immunity
16 of 100
Diagnostic Tools: Molecular Probes for the Detection of Biological Aldehydes
17 of 100
A Generalized Approach to Deliver Functionalized Isoindolines in Macrocycles
18 of 100
Developing Transition Metal Catalysts that Incorporate Redox-Active Ligand Frameworks for Sustainable Catalysis
19 of 100
Development of New Diaryl Diazo Compounds and the Study of their application in C-H Functionalization Chemistry
20 of 100
Development of New Diaryl Diazo Compounds and the Study of their application in C-H Functionalization Chemistry
21 of 100
DNA mechanocapsules: Force responsive tetrahedral DNA nanostructures with modular cargo delivery for targeting mechanical phenotypes of diseases
22 of 100
Metal Catalyst Methodology Development towards Carbon-Oxygen Bond Formation: Synthesis of Vinyl Ethers and Vinyl Esters
23 of 100
The Development of Planar Chiral Indenyl Catalysts and the Progress Towards Synthesis of the Western Macrocycle of Darobactin A
24 of 100
Group IX Metal-Catalyzed C–H Activation Towards the Development of New Synthetic Strategies
25 of 100
Natural Product Inspired Complementary Approaches to Counter Antimicrobial Resistance: Synthetic and Biological Investigations of Antibacterial Small Molecules
26 of 100
An Investigation on the Diastereoselectivity of α-Methylstyrene Cyclopropanations Catalyzed by Dirhodium (II) Catalysts
27 of 100
Synthesis of Novel Nucleotide Tenofovir/Lamivudine Prodrug Conjugates for treatment of Human Immunodeficiency Virus and Hepatitis B
28 of 100
Synthesis and Evaluation of Novel Phenyl-Adamantane Dirhodium Catalyst for C-H Functionalization
29 of 100
New Advances in Asymmetric Cyclopropanation and Drug Discoveries Using Dirhodium(II) Tetracarboxylates
30 of 100
Asparagine and Glutamine Bioconjugation
31 of 100
Synthesis of alkyl analogues of 1,4-dihydropyridine for developing novel treatment against chemoresistance in prostate cancer
32 of 100
Carboxylation of C(sp2) Bromides Enabled by Metallophotoredox Dual Catalysis and Sodium Formate
33 of 100
Computational Modeling of Oxyradical and Metal-Oxo Reactivity and Selectivity in Hydrogen Atom Transfer Reactions
34 of 100
Triazene Coarctate Cyclization for the Synthesis of Fluorescent Cyclic Peptides
35 of 100
Overcoming Antibacterial Resistance through Synthesis of Small Molecules Targeting Efflux Mechanisms
36 of 100
Overcoming the Limitations of Rhodium-Catalyzed Asymmetric Cyclopropanation and Other Adventures in Strained Ring Synthesis
37 of 100
Catalytic Process for Epoxide Ring-Opening with Terminal Alkynes for Carbon-Carbon Bond Formation
38 of 100
Novel Quaternary Ammonium Compounds Derived from the Antimicrobial Natural Product Ianthelliformisamine C
39 of 100
Cu- and Pd-Catalyzed a-Hydroxycyclopropanol Ring Opening Reactions: Electrophilic Trappings to 3-Furanones, and Carbonylation to 4-Ketovalerolactones.
40 of 100
Radical Reactivity via Transient Carbon Dioxide Radical Anion (CO2•−)
41 of 100
Design and Synthesis of Chemical Modulators for Altered Activity of Nuclear Receptor Liver Receptor Homolog-1 and Synthesis of Spirocyclic Piperidines via Radical Hydroarylation
42 of 100
Chemo and Site Selective Modification of Proteins and Chemical Tools for Studying Mono-Methyl Lysine (Kme)
43 of 100
Developing Chemical Tools for Selective Peptide Modification
44 of 100
Studies in Small Molecule Drug Discovery: Part I. Synthesis of Novel Nucleoside-Based Antivirals to Treat Hepatitis C; Part II. Validation and Implementation of a Machine Learning Algorithm to Create a Safer Kinase Inhibitor as a Potential First-in-Class Antiparkinsonian Agent
45 of 100
Membranes & Metals: Bacterial Targets to Fight Antibiotic Resistance
46 of 100
Exploration of Bilingual Peptide Nucleic Acids
47 of 100
Development of Chemical Methods for Labeling Monomethyl Lysine Post-Translational Modification and Serine and their Applications.
48 of 100
A Three-Pronged Approach to Combatting Antibiotic Resistance
49 of 100
Synthesis and Biological Investigation of Membrane-targeting Antimicrobials
50 of 100
Synthesis and Biological Investigation of Natural Product-Inspired Antimicrobial Compounds
51 of 100
Fibrinogen and Clotting Characterization in COVID-19 Patients
52 of 100
Synthetic Investigations into Small Molecules with Antibacterial Potential
53 of 100
Site-Selective and Enantioselective C-H Functionalization of Unactivated C–H Bonds in the Presence of Nitrogen Functionality
54 of 100
Synthesis of Novel EP2 Prostaglandin Antagonists for Optimal Blood-Brain Barrier Permeation as Radioligands
55 of 100
Computational Development of Macrocyclic Drug Hits and Synthetic Strategy towards Peptide Macrocyclization
56 of 100
Leveraging Chemical Tools to Target Bacterial Membranes and Combat Antimicrobial Resistance
57 of 100
Asymmetric Rhodium(II)-Carbene C-H Functionalization: A Complementary Tool To Synthetic Disconnection Strategies
58 of 100
Glyoxal-based Caging of Nucleoside Reverse Transcriptase Inhibitors for the Treatment of Viral Infections
59 of 100
Total synthesis and biological investigations of natural product inspired antimicrobials
60 of 100
C-H Functionalization Inspired Total Synthesis and New Donor/Acceptor Carbenes for Asymmetric C-H Functionalization
61 of 100
Leveraging Organic Synthesis to Disrupt and Understand Essential Bacterial Processes
62 of 100
Practical Application and In Situ Kinetic Studies of Dirhodium(II) Tetracarboxylate Catalyzed Carbene Reactions
63 of 100
Targeting Bacterial Tolerance and Resistance with Small Molecules
64 of 100
Design, Synthesis, and Utility of Group IX Metal Catalysts for C–H Functionalization
65 of 100
Dearomative Photocatalytic Hydroalkylation and Lipophilic Prodrugs
66 of 100
A Tale of Two Chemistries: Dynamics of Delay-Coupled Belousov-Zhabotinsky Oscillators; TrkB Activators: A Review; Synthesis of TrkB Agonists
67 of 100
Cobalt Catalyzed Intramolecular Cyclization of Acyclic Alkenols for Polycyclic Ether Synthesis
68 of 100
EXPANDING THE SCOPE AND APPLICATION OF N-SULFONYL-1,2,3-TRIAZOLES AS ALTERNATE PRECURSORS TO DONOR/ACCEPTOR RHODIUM CARBENES
69 of 100
Arene Dearomatization via Radical Hydrofunctionalization
70 of 100
Design and Synthesis of a PD-L1 Radioligand for Diagnostic Imaging and Development and Optimization of a Potent Liver Receptor Homolog-1 Agonist
71 of 100
The Iterative Design of Aptamer-Functionalized Membranes to Enable Detection, Sequestration, and Recovery of Small-Molecule Compounds
72 of 100
Intercepting Photochemically Generated Aminoalkyl and Aryl Radical Intermediates to Access Complexity Quickly
73 of 100
Developing First-Row Transition Metal Complexes for Green Catalytic C–H Activation and Oxidations
74 of 100
GluN2C/D subunit selective antagonist for NMDARs: 997 Series
75 of 100
Optimization of Rh2(S-TPPTTL)4 Through Ligand Diversification
76 of 100
Unusual Paradigms in Selective Synthesis: Part 1: Toward the Synthesis of Racemic and Enantioenriched HIOC; Part 2: Fluorinated Alcohols: Powerful Promoters for the Ring-Opening Reactions of Epoxides with Carbon Nucleophiles
77 of 100
Probing Bacterial Mechanisms via Small Molecule Antibiotics
78 of 100
Design and Synthesis of New Liver Receptor Homolog-1 Modulators and Probes
79 of 100
The Development and Mechanistic Studies of Group(IX)Cp*-Catalyzed Allylic C–H Functionalization Reactions Proceeding via a π-allyl Intermediate
80 of 100
Studies Towards the Synthesis of Malagasy Alkaloids, and Development and Applications of Regio- and Enantioselective Group IX Metal-Catalysed Reactions
81 of 100
Structural Requirements of the Sulfonyl Prolinate Ligands for Dirhodium Catalysis
82 of 100
Computational and Experimental Studies of Selective Rhodium-Catalyzed Allylic C–H Functionalization through π-Allyl Intermediates and Computational Development of Macrocycle Leads for Undruggable Targets
83 of 100
Harnessing the Dual Nature of Peptide Nucleic Acids
84 of 100
Broadening the applications of rhodium donor/acceptor carbene mediated C–H functionalization
85 of 100
Allylic C-H Arylation, Enantioselective Catalyst Development, and Enantioselective Allylic C-H Amidation
86 of 100
Exploring the Influence of Dirhodium Catalyst Structure on the Regio- and Stereoselectivity Properties of Donor/Acceptor Carbenes
87 of 100
Development and Applications of a New Dirhodium(II) Tetracarboxylate Catalyst and Asymmetric Cyclopropanation of Heterocyclic Compounds
88 of 100
Investigation of the Bridgehead Substituent of the Leading LRH-1 Agonists
89 of 100
Radical Conjugate Addition of N-Heterocycles and Tertiary Amines
90 of 100
Synthetic Applications of Dirhodium(II) Catalysis
91 of 100
Development and Optimization of Monosubstituted and Disubstituted Alkene Synthesis for Future Intramolecular Alkene Hydroalkoxylation Reactions
92 of 100
Modification of Quorum Quenching Analogs from Schinus terebinthifolia Fruit Extract
93 of 100
Synthesis of a Click-Compatible Phenylacrylamide to Probe A-to-I RNA Editing
94 of 100
Synthesis of a novel C-nucleoside prodrug for treatment of Hepatitis B
95 of 100
Allylic C-H Functionalization Studies on Allylbenzene Derivatives
96 of 100
Development of Intermolecular Couplings of Aryl Radical Species with Olefins
97 of 100
Reductive Processes Enabled by Photoredox for the Synthesis and Modification of Pharmaceutically Relevant Molecules
98 of 100
Synthesis, Structure-Activity Relationship, and Biological Evaluation of Subunit-Selective NMDA Receptor Modulators
99 of 100
Carolacton and Honokiol: using natural product inspiration to target the oral microbiome
100 of 100